SRPK inhibitor
Catalog No. S21-901
| Catalog No. | Pack Size | Price (USD) | |
|---|---|---|---|
| S21-901-05 | 5 mg | $105 | |
| S21-901-25 | 25 mg | $410 | |
| S21-901-BULK | BULK | Contact Us |
Overview:
Serine arginine protein kinase (SRPK) 1 inhibitor (Ki = 0.89 µM)1. Inhibits SRPK2 at higher concentrations. Does not significantly inhibit other SRPKs such as CLK1 and CLK4, or other classes of SR kinases.
References:
1. T Fukuhara et al. Proc. Natl. Acad. Sci. USA 2006 103:11329
2. MV Gammons et al. Invest. Ophthalmol. Vis. Sci. 2013 54:5797
3. MV Gammons et al. Br. J. Cancer 2014 111:477
CAS Registry Number:
218156-96-8
Molecular Formula:
C18H18F3N3O
Appearance:
White powder
Molecular Weight:
349.4
Purity:
>98% (TLC); NMR (Conforms)
Solubilization:
May be dissolved in DMSO (40 mg/ml) or ethanol (25 mg/ml)
Aliases:
N-[2-(1-Piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamide
Storage and Stability:
Store desiccated as supplied at -20oC temperature for up to 2 years. Store solutions at -20oC for up to 1 month.
Molecular Structure:
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There are no related publications available for this product.
Cancer, Inflammation, Neurobiology, Ser/Thr Kinases
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